Smit et al. 2019

Population pharmacokinetics of vancomycin in obesity: Finding the optimal dose for (morbidly) obese individuals

British Journal of Clinical Pharmacology · 10.1111/bcp.14144

Structure

A three-compartment model, driven by weight and age.

Study population

Obese, General and Mixed patients — Netherlands and Europe. Fitted to 28 patients and 326 concentration observations.

Covariate As reported
Age 35.2 (20–55) yr
Weight 104.3 (60–234.6) kg
BMI 37.9 (20.4–65.7) kg/m²
CrCl 135.5 ± 39 mL/min
SCr 0.72 (0.41–1.01) mg/dL

Reported as the source publication gives them — mean ± SD, or median with range or interquartile range.

Equations

The model's structural parameters as Chorus implements them.

CL=5.72(Weight70)0.535CL = 5.72 \cdot \left(\frac{Weight}{70}\right)^{0.535}V1=16.7(1+0.0136(Age36.5))V_1 = 16.7 \cdot (1 + 0.0136 \cdot (Age - 36.5))V2=6.98Weight70(1+0.0136(Age36.5))V_2 = 6.98 \cdot \frac{Weight}{70} \cdot (1 + 0.0136 \cdot (Age - 36.5))V3=19.5V_3 = 19.5Q2=15.8Q_2 = 15.8Q3=5.21Q_3 = 5.21
LaTeX source
CL = 5.72 \cdot \left(\frac{Weight}{70}\right)^{0.535}
V_1 = 16.7 \cdot (1 + 0.0136 \cdot (Age - 36.5))
V_2 = 6.98 \cdot \frac{Weight}{70} \cdot (1 + 0.0136 \cdot (Age - 36.5))
V_3 = 19.5
Q_2 = 15.8
Q_3 = 5.21

Implementation notes

Three-compartment model. BMI-dependent IIV on clearance. No renal function covariates - developed in patients with normal renal function only.

Simulation settings

Models

selected

Dose candidates (mg)

Interval candidates (h)

Demographics

Physical characteristics.

kg
cm
yr